(1215-D) Affinity Selection-Mass Spectrometry HTS Applied to Challenging Drug Targets.
Tuesday, February 6, 2024
2:00 PM – 3:00 PM EST
Location: Exhibit Halls AB
Abstract: HTS by Affinity Selection-Mass Spectrometry enables rapid ID of mass-verified ligands with desired functional actions on proteins of interest. Comprising advanced data analysis, highly sensitive detection, and precise automation, these systems are typically custom-evolved and perfected in industry laboratories. Outsourcing to specialized providers with complementary automated systems has efficiently addressed several needs across a diverse early discovery pipeline. This strategy and its output of lead-like hits with potent functional activity will be described in the context of platforms' respective technical features.